Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04527
Ion Channel
Glutamate receptor ionotropic subunit NMDA 1
Peptide Function
Antagonist
Gene Name
Grin1
Activity Data (nM)
IC50
171 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GEXXLQXNQXLXRXKSN
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
[Conotoxin GV; Conotoxin G V; 93438-65-4; Sleeper peptide; Snail sleeper peptide; Conantokin-G; Conantokin G; UNII-32CFR9L3TD; CGX-1007; 32CFR9L3TD; Conotoxin G V;GEXXLQXNQX LIRXKSN; DTXSID10896916; AKOS024457994; NS00075388]
Peptide Species
Conus geographus (Geography cone) (Nubecula geographus)
Peptide Name
Conantokin-G
CAS Number
93438-65-4
Experimental Conditions
pH
pH 7.5
Holding Potential (mV)
Not specified
Temperature
30 °C
Test Method
Binding assay
Test Species
Not specified
Binding Information
Binding Site
Extracellular domain
Binding Site Residue
GIy binding site
Ion Channel Information
Gene Abbreviation (ABB)
i-GluRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available